Transporters as Targets for Drugs

1. Overview: Transporters as Targets for Drug Discovery
Matilda Bingham, Susan Napier

2. Membrane Transporters: Structure, Function and Targets for Drug Design
Aina W. Ravna, Georg Sager, Svein G. Dahl, Ingebrigt Sylte

3. Design of Monoamine Reuptake Inhibitors: SSRIs, SNRIs and NRIs
Gavin A. Whitlock, Mark D. Andrews, Alan D. Brown, Paul V. Fish, Alan Stobie, Florian Wakenhut

4. Atypical Dopamine Uptake Inhibitors that Provide Clues About Cocaine's Mechanism
at the Dopamine Transporter
Amy Hauck Newman, Jonathan L. Katz

5. The Design, Synthesis and Structure–Activity Relationship of Mixed Serotonin,
Norepinephrine and Dopamine Uptake Inhibitors
Zhengming Chen, Ji Yang, Phil Skolnick

6. Molecular Imaging of Transporters with Positron Emission Tomography
Gunnar Antoni, Jens Sörensen, Håkan Hall

7. Pharmacology of Glutamate Transport in the CNS: Substrates and Inhibitors of Excitatory
Amino Acid Transporters (EAATs) and the Glutamate/Cystine Exchanger System x
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Richard J. Bridges, Sarjubhai A. Patel

8. Glycine Transporters and Their Inhibitors
Robert Gilfillan, Jennifer Kerr, Glenn Walker, Grant Wishart

Keywords: Chemistry, Medicinal Chemistry, Pharmacology/Toxicology, Organic Chemistry, Molecular Medicine