Iverson, Suzanne L.
Metabolite Safety in Drug Development
• Reviews the analytical techniques and experimental designs critical for metabolite studies
• Covers methods including chirality, species differences, mass spectrometry, radiolabels, and in vitro / in vivo correlation
• Discusses target pharmacology, in vitro systems aligned to toxicity tests, and drug-drug interactions
• Includes perspectives from authors with firsthand involvement in industry and the study of drug metabolites, including viewpoints that have influenced regulatory guidelines
Keywords: Drug metabolism; drug metabolites; metabolite safety; metabolite studies; drug development; target pharmacology; toxicity tests; drug-drug interactions; drug candidate selection, Pharmacology & Pharmaceutical Medicine, Analytical Chemistry, Pharmacology & Pharmaceutical Medicine, Analytical Chemistry
- Editor
- Iverson, Suzanne L.
- Smith, Dennis A.
- Publisher
- John Wiley and Sons, Inc.
- Publication year
- 2016
- Language
- en
- Edition
- 1
- Page amount
- 352 pages
- Category
- Natural Sciences
- Format
- Ebook
- eISBN (ePUB)
- 9781118949672
- Printed ISBN
- 9781118949658