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Valle, Susan Del

Peptides for Youth

Valle, Susan Del - Peptides for Youth, ebook

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ISBN: 9780387736570
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Table of contents

1. Dynamic Combinatorial Assembly of Peptide-Rhenium Coordinates: Application to the Selection of hCyp-18 inhibitors from a Library of 12 × 16 Components
C. Dugave, C. Clavaud, J. Le Gal, R. Thai, M. Moutiez

2. Dynamic Combinatorial Assembly of Peptide-Rhenium Coordinates: Coordination Chemistry for Generating New Analogs of hCyp-18 Ligands
C. Clavaud, J. Le Gal, R. Thai, M. Moutiez, C. Dugave

3. Oxorhenium-Mediated Cyclization and Self-Assembly of Peptides: A Combinatorial Approach for the Selection of New Ligands of the Human Cyclophilin hCyp-18
C. Clavaud, M. Heckenroth, C. Stricane, M-A. Lelait, A. Ménez, C. Dugave

4. Thieno[3,2-e]diazepinediones and 3-Thienylimidazolidinediones Syntheses: Regio-Controlled Ring Opening of Thiaisatoic Anhydride by α-Amino Acids.
Yann Brouillette, Vincent Lisowski, Jean Martinez

5. Solid-Phase Synthesis of Phosphinic Dipepetide Isosteres and β Amino Acids via Activated N-Terminal Acrylamides
Florian Manzenrieder, Horst Kessler

6. Parallel Solid-Phase Synthesis of Macrocyclic Peptidomimetics Using Ru-Catalyzed Ring-Closing Metathesis and a New Application of Cross Metathesis
Sylvie Beaubien, Hamid R. Hoveyda, Martin Vézina, Éric Marsault, Hugo Tremblay, Laurence Foucher, Kamel Benakli

7. High Throughput Solid Phase Parallel Synthesis of Macrocyclic Peptidomimetics
E. Marsault, H. R. Hoveyda, M. L. Peterson, R. Gagnon, M. Vézina, J.F. Pinault, A. Landry, C. Saint-Louis, L. G. Ouellet, S. Beauchemin, K. Benakli, S. Beaubien, M. Brassard, Z. Wang, M. Champagne, F. Galaud, N. Fortin, D. Fortin, V. Plourde, M. Ramaseshan, S. Bhat, F. Bilodeau, D. Lonergan, R. Lan, S. Li, G. Berthiaume, L. Foucher, X. Peng, Y. Dory, P. Deslongchamps

8. Development of an Efficient Solid-Phase Synthetic Methodology to Construct a Combinatorial Library of a Potent HDAC Inhibitor
Salvatore Di Maro, Jung-Mo Ahn

9. A Novel Hydrogel Functionalized with Specific Peptidomimetic Ligands for 2-D and 3-D Cell Culture
Juntao Luo, Ekama Onofiok, Changying Shi, Ruiwu Liu, Kit S. Lam

10. Application of the “Libraries from Libraries” Concept to “One-bead One-compound” Combinatorial Chemistry
Joseph C. Kappel, Yi C. Fan, Kit S. Lam

11. An Appreciation of the Scientific Life and Achievements of Bruce Merrifield
Alexander R. Mitchell

12. The “Bip Method” for Spectroscopic Assignment of the Absolute Configuration of the Spin-Labelled, Cyclic β2,3-Amino Acids β-TOAC and POAC
Karen Wright, Laurencev Dutot, Anne Gaucher, Michel Wakselman, Jean-Paul Mazaleyrat, Cristina Peggion, Fernando Formaggio, Claudio Toniolo

13. Enzyme Mechanism and Function of a Novel Plant PDI Involved in the Oxidative Folding of Cystine Knot Defense Peptides
Christian W. Gruber, Maša Čemažar, Marilyn A. Anderson, David J. Craik

14. Biosynthesis of Siderophore-Peptides, A Class of Potent Antimicrobial Peptides from Enterobacteria, Requires Two Precursors
Gaëlle Vassiliadis, Jean Peduzzi, Delphine Destoumieux-Garzón, Séverine Zirah, Xavier Thomas, Sylvie Rebuffat

15. Post-Translational Modification and folding of A Lasso-Type Gene-Encoded Antimicrobial Peptide Require Two Enzymes only in Escherichia coli

Sophie Duquesne, Delphine Destoumieux-Garzón, Séverine Zirah, Thomas A. Knappe, Christophe Goulard, Jean Peduzzi, Mohamed A. Marahiel, Sylvie Rebuffat

16. Synthesis and 3D-Structure of Conformationally Controlled Nucleo-Peptides
Piero Geotti-Bianchini, Marco Crisma, Cristina Peggion, Alberto Bianco, Fernando Formaggio

17. Mixing Urea and Amide Bonds: Synthesis and Self-Organization of New Hybrid Oligomers
Lucile Fischer, Gersande Lena, Jean-Paul Briand, Claude Didierjean, Gilles Guichard

18. Optimizing the Fold Stability of Miniprotein Sequences
D. Victoria Williams, Jasper C. Lin, Brandon L. Kier, Niels H. Andersen

19. Antimicrobial Peptides Chelating Lanthanide Ions: the Case of Trichogin GA IV Analogues and Terbium(III)
Mariano Venanzi, Emanuela Gatto, Lorenzo Stella, Gianfranco Bocchinfuso, Antonio Palleschi, Fernando Formaggio, Claudio Toniolo

20. Spectroscopic Characterization of the Fully-Extended, Planar, Peptide 2.05-Helix Based on Chiral, Cα -Ethylated, α-Amino Acids
Claudio Toniolo, Marco Crisma, Fernando Formaggio, Alessandro Moretto, Cristina Peggion, Bernard Kaptein, Quirinus B. Broxterman

21. Monitoring Peptide Folding by Time-Resolved Spectroscopies: the Effect of a Single Gly to Aib Susbtitution
Mariano Venanzi, Emanuela Gatto, Gianfranco Bocchinfuso, Antonio Palleschi, Lorenzo Stella, Chiara Baldini, Fernando Formaggio, Claudio Toniolo, Basilio Pispisa

22. First Homo-Peptides Undergoing a Reversible 310-Helix to α-Helix ransition
Alessandro Moretto, Marco Crisma, Fernando Formaggio, Claudio Toniolo, Ling Wu, Timothy A. Keiderling, Bernard Kaptein, Quirinus B. Broxterman

23. Molecular Modeling Approach to Achieving Erythropoietin Mimetic Peptides
Yanfeng Qi, Xuefeng Gao, Liping Wang, Wei Li

24. Conformation Analysis of Parathyroid Hormone Residues Critical for Bioactivity
Zhanna Potetinova, Feng Ni, Manghaiko Mayele, Ping Xu, Gordon E. Willick

25. Light-Switchable Folding/Unfolding of the Collagen Triple Helix with Azobenzene-Containing Model Peptides
Ulrike Kusebauch, Lisa Lorenz, Sergio A. Cadamuro, Hans-Jürgen Musiol, Martin O. Lenz, Christian Renner, Josef Wachtveitl, Luis Moroder

26. Structural Studies of Parathyroid Hormone Analogue with C-Terminal Aldehyde Function
Zhanna Potetinova, Feng Ni, Ping Xu, Gordon E. Willick

27. Synthesis and Conformational Studies of Novel, Side-Chain Protected, L-(aMe)Ser Homo-Peptides
Fernando Formaggio, Cristina Peggion, Claudio Toniolo, Bernard Kaptein, Quirinus B. Broxterman, Minghong Ni, Laura Muzi, Alma Dal Pozzo

28. Introduction of N-alkyl Residues in Proline-rich Peptides: Effect on SH3 Binding Affinity and Peptide Conformation
Paolo Ruzza, Chiara Rubini, Giuliano Siligardi, Rohanah Hussain, Andrea Calderan, Andrea Guiotto, Luca Cesaro, Anna M. Brunati, Arianna Donella-Deana

29. Thermodynamic Stability And Native-State Dynamics Of Porcine Pancreatic Phospholipase A2 Studied By 1H NMR Spectroscopic Measurements
Carmen Mrestani-Klaus, Knut Kölbel, Renate Ulbrich-Hofmann

30. The amyloidogenic domains of the human serum amyloid A protein -New Insights-
Emanuel Perugia, Elena Monticelli, Sarah Rubinraut, Aviva Kapitkovsky, Mati Fridkin

31. Quantitating Amino Acid β-Strand Preferences, Turn Propensities and Cross-Strand Interactions in a Designed Hairpin Peptide
Kelly N. Huggins, Niels H. Andersen

32. Determinants of fold stabilizing aromatic-aromatic interactions in short peptides
Lisa A. Eidenschink, Brandon L. Kier, Niels H. Andersen

33. Spectroscopic analysis of synthetic PrP helix2-binding peptide constructs
Luisa Ronga, Pasquale Palladino, Raffaele Ragone, Jean Martinez, Ettore Benedetti, Filomena Rossi, Muriel Amblard

34. Unique Role of Clusters of Electrostatic Attractions in Controlling the Stability of Two-stranded α-Helical Coiled-Coils
J. Paul Kirwan, Stan C. Kwok, Susanna McReynolds, Janine Mills, David Osguthorpe, Robert S. Hodges

35. The Energetics of Weakly Polar Interactions in Model Tripeptides
József Csontos, Richard F. Murphy, Sándor Lovas

36. Peptidomimetic Ligands for the Tandem SH2 Domain of the Syk Protein Involved in Signal Transduction
Joeri Kuil, Loek T. M. van Wandelen, Nico J. de Mol, Rob M. J. Liskamp

37. Subtilisin Kexin Isozyme-1 (SKI-1): Production, purification, inhibitor design and biochemical applications
Dayani Mohottalage, Natalie Goto, Ajoy Basak

38. Effects of Antifreeze Protein Fragments on the Properties of Model Membranes
Hagit Kun, Gerardo Byk, Yitzhak Mastai

39. Fluorogenic Cyclooctapeptides and Metal Ion Sensing
Maria Ngu-Schwemlein, Liliana Garcia, Kshawna Askew

40. The Impact of Aromatic Residues on the Tertiary Fold of Avian Pancreatic Polypeptide
Nicholas Y. Palermo, József Csontos, Richard F. Murphy, Sándor Lovas

41. An Efficient Protocol for On-Resin, Vicinal Disulfide Formation: Applications to Thioredoxin Reductase
Stevenson Jr Flemer, Robert J. Hondal

42. Potent and selective peptide agonists for human melanocortin receptor 5
Maria A. Bednarek, Tanya MacNeil, Rui Tang, M. Angeles Cabello, Marta Maroto, Ana Teran

43. Synthesis of a library of Ψ-stylostatins with potential antibacterial activity
Carlos López, Montse Cruz, Javier Sánchez-Cespedes, Anna Diez

44. Mimicking natural globular structures with rigid scaffolds based on adamantane
Nadine Pannier, John V. Frangioni, Wolfgang Maison

45. Discovery and Optimization of a TRAIL R2 Agonist for Cancer Therapy
Yvonne M. Angell, Ashok Bhandari, M. Nuria De Francisco, Brian T. Frederick, Jennifer M. Green, Karen Leu, Kerstin Leuther, Reuben Sana, Peter J. Schatz, Erik A. Whitehorn, Kathy Wright, Christopher P. Holmes

46. Novel reactive site loop derived mini-serpin inhibitors of recombinant Proprotein Convertase 4
Ajoy Basak, Nausheen Shervani, Maria Kolajova, Shalini Cherla, Sarmistha Basak

47. Enzymatic ligation of peptides, peptide nucleic acids and proteins by means of sortase A
Stephan Pritz, Yvonne Wolf, Oliver Kraetke, Jana Klose, Michael Bienert, Michael Beyermann

48.
N-Methylated Cyclic Pentapeptides as Template Structures
Jayanta Chatterjee, Oded Ovadia, Chaim Gilon, Amnon Hoffman, Dale Mierke, Horst Kessler

49. Cyclic Dimers Of C-terminal γ2-MSH Analogs As Selective Antagonists Of The Human Sensory Nerve-Specific Receptor (SNSR-4)
Ralf Schmidt, Joanne Butterworth, Dajan O'Donnell, V. Santhakumar, Mirek Tomaszewski

50. Structure-Function Relationship Study of Parathyroid Hormone (1–11) Analogues Containing D-AA
A. Caporale, N. Fiori, E. Schievano, A. Wittelsberger, S. Mammi, M. Chorev, E. Peggion

51. Selective enzymatic hydrolysis of C-terminal tert-butyl esters of peptides
Carmen G. Boeriu, Ivo F. Eggen, Dirk-Jan van Zoelen, Gilbert H. Bours

52. Peptide Ligation via the In-Situ Transformation of an Amide into a Thioester at a Cysteine Residue
Toru Kawakami, Saburo Aimoto

53. Facile Synthesis of Glucagon-Like Peptide-1 (GLP-1) Mimetics
Sun-Young Han, Martin Beinborn, Jung-Mo Ahn

54. Synthetic Peptide Vaccines: The Quest to Develop Peptide Vaccines for Influenza, HIV and Alzheimer's Disease
Elisabetta Bianchi, Paolo Ingallinella, Marco Finotto, Joseph Joyce, Xiaoping Liang, Michael D. Miller, Gene G. Kinney, Gennaro Ciliberto, John W. Shiver, Antonello Pessi

55. Rational Design of Peptidomimetics for Class B GPCRs: Potent Non-Peptide GLP-1 Receptor Agonists
Jung-Mo Ahn, Sun-Young Han, Eunice Murage, Martin Beinborn

56. The depsipeptide technique for the solid phase peptide synthesis: from stepwise assembly to segment condensation
Irene Coin, Peter Schmieder, Michael Bienert, Michael Beyermann

57. A Novel Method for the Preparation of Peptide Thioester and its Application to Glycoprotein Synthesis
Hironobu Hojo, Yuko Onuma, Yuri Akimoto, Yuko Nakahara, Yoshiaki Nakahara

58. Synthesis of 4-arylmethyl-L-histidine analogues for structure-activity studies of position 10 of CGRP
D. David Smith, Michael Mao, Hayley Young, Martin Hulce

59. Solid-phase synthesis of dipeptidic and pseudo-dipeptidic potential NOS inhibitors through a side-chain anchoring approach
Youness Touati-Jallabe, Abdallah Hamzé, Gilbert Bergé, Claudia Verna, Anne-Dominique Lajoix, Pierre Fulcrand, Jean Martinez, Jean-François Hernandez

60. Further Development of New Deprotection Chemistry for Cysteine and Selenocysteine Side Chain Protecting Groups
Alayne L. Schroll, Robert J. Hondal

61. A New Synthesis of (+)-Negamycin and Its Derivatives as a Potential Therapeutic Agent for Duchenne Muscular Dystrophy Treatment
Yoshio Hayashi, Shigenobu Nishiguchi, Magne O. Sydnes, Thomas Regnier, Jun-ya Hasegawa, Takahiro Katoh, Tetsuya Kajimoto, Manabu Node, Yoshiaki Kiso

62. Design and Synthesis of Backbone Cyclic Phosphopeptides: The IκB Model
Nir Qvit, Ada Hatzubai, Deborah E. Shalev, Yinon Ben-Neriah, Chaim Gilon

63. Synthesis of modified and hybrid protein derived biopolymers
Jimmy J. Weterings, Selina Khan, Jan W. Drijfhout, Ferry Ossendorp, Herman S. Overkleeft, Gijsbert A. van der Marel, Dmitri V. Filippov

64. SPPS of the Natural Product Chitinase Inhibitor Argifin: Library Generation and Biological Evaluation
Mark J. Dixon, Ole A. Andersen, Daan M. F. van Aalten, Ian M. Eggleston

65. Development of Chemokine Receptor CXCR4 Antagonists Using Bio-mimetic Strategy
Hirokazu Tamamura, Tomohiro Tanaka, Hiroshi Tsutsumi, Nami Ohashi, Kenichi Hiramatsu, Takanobu Araki, Akio Ojida, Itaru Hamachi, Zixuan Wang, Stephen C. Peiper, John O. Trent, Satoshi Ueda, Shinya Oishi, Nobutaka Fujii

66. Chemical Synthesis of the N-Terminal Cysteine-Rich Domain of Human OX40
Tami L. Raguse, Steven C Pomerantz, Jennifer F. Nemeth, Jinquan Luo, Audrey E. Baker, Jian Li, Diane Deriggi, Raymond Sweet, Marian Kruszynski

67. Stereoselective Synthesis of Peptidomimetics Based on Acid-catalyzed Ring-opening of β-Aziridinyl-α,β-enoates
Hirokazu Tamamura, Tomohiro Tanaka, Hiroshi Tsutsumi, Koji Nemoto, Satoko Mizokami, Nami Ohashi, Shinya Oishi, Nobutaka Fujii

68. Development of a small molecule peptidomimetic affinity Ligand for efficient purification of the large protein Factor VIII
Sebastian Knör, Burkhardt Laufer, Alexey Khrenov, Abdellah Benhida, Sabrina C. Grailly, Nathalie Beaufort, Viktor Magdolen, Charlotte A. E. Hauser, Evgueni L. Saenko, Jean-Marie R. Saint-Remy, Horst Kessler

69. Expression and Characterization of Recombinant S2 Subunit of SARS-coronavirus S Fusion Protein
Zhe Yan, Kathryn V. Holmes, Robert S. Hodges

70. Synthesis of Biotinyl-TN14003, Anti-HIV Peptide Amide
H. Nedev, H. U. Saragovi

71. Making double-minded peptides strong-willed? The side chain impact on the backbone conformation of N-methylated cyclic pentapeptides
Burkhardt Laufer, Jayanta Chatterjee, Andreas O. Frank, Horst Kessler

72. Deprotection of N

in
-Formyl Group on Tryptophan by Application of New Reagent, 1,2-dimethylethylendiamine in Aqueous Solution
Takenao Odagami, Yuji Kogami, Hiroyuki Kouji, Yuko Tsuda, Yoshio Okada

73. Racemization-free segment condensation based on the O-acyl isopeptide method: Toward a chemical protein synthesis on solid support
Taku Yoshiya, Youhei Sohma, Yoshio Hamada, Tooru Kimura, Yoshio Hayashi, Yoshiaki Kiso

74. Optimized Coupling Protocols for the Incorporation of Cys Derivatives during Fmoc-SPPS
Guenther Loidl, Fritz Dick, Monika Mergler, Ralph O. Schoenleber

75. Further studies on peptide synthesis at high temperature
Carina Loffredo, Nilson A. Assunção, M. Terêsa M. Miranda

76. Preparation of C-terminal modified peptides through alcoholysis and thiolysis mediated by metal ions
Patrícia B. Proti, M. Terêsa, M. Miranda

77. Synthesis and Biological Activity of Amino Acid Esters of Acyclovir
Ivanka Stankova, Tatyana Dzimbova, Stoyan Shishkov

78. Poly-(ProΨ[CH(OAc)CH2]Aib)3 a Protected Trimer of Pro-Aib Hydroxyethylene Isosteres
T. Lama, G. Fridkin, W. D. Lubell

79. Fast Conventional Synthesis of Human ß-Amyloid (1–42) on the Symphony® and Prelude™
German Fuentes, Christina Hood, Jae H. Park, Hirendra Patel, Karen Page, Mahendra Menakuru

80. Side chain-to-Side chain Cyclization by Intramolecular Click Reaction - Building Blocks, Solid Phase Synthesis and Conformational Characterization
Sonia Cantel, Jose A. Halperin, Michael Chorev, Mario Scrima, Anna M. D'Ursi, Jay J. Levy, Richard D. DiMarchi, Alexandra Le Chevalier, Paolo Rovero, Anna M. Papini

81. An Efficient Approach to Synthesize Multiple Peptides with Carboxyl C-termini
Koichiro Hayashi, Sylvia Chen, Paul Opare-Addo, Ashok Khatri

82. Synthesis and Biological Activity of Novel α-Conotoxin Analogues Incorporating Substituted Proline Derivatives
Christopher J. Armishaw, Anders A. Jensen, Christian Skonberg, Tommy Liljefors, Kristian Strømgaard

83. Application of Triethylsilane and Palladium-Charcoal-Induced Reductions in the Synthesis of Fmoc-Glutamic Acid Analogues
Pijus K. Mandal, John S. McMurray

84. Synthesis of pyrrolo[3,2-e][1,4]diazepin-2-ones as potential γ-turn mimetics
Philippe Deaudelin, William D. Lubell

85. Improvements in the Chemical Synthesis of Insulin-Like Peptides
Panagiota Tsetseni, Aggeliki Karkantzou, Spyros Markos, Kostas Barlos, Dimitrios Gatos, Kleomenis Barlos

86. Design And Parallel Synthesis Of New Bicyclic Small Molecules For Targeting The Melanocortin Receptors
Byoung J. Min, Alexander V. Mayorov, Minying Cai, Erin Palmer, Victor J. Hruby

87. Fully Automated Fast Fmoc Synthesis and On-Resin Disulfide Bridge Formation with Pseudoproline Dipeptides on the Prelude™ [1]
Karen Page, Jae H. Park, Christina A. Hood, Hirendra Patel, German Fuentes, Mahendra Menakuru

88. Efficient Synthesis of Protected L-Phosphonophenylalanine (Ppa) Derivatives Suitable for Solid Phase Synthesis
Satendra S. Chauhan, A. Varshney, B. Verma, Michael W. Pennington

89. ALLESSAN CAP - A Highly Versatile And Affordable Coupling Agent
Richard Amitrano, Peter Koch, Marita Neuber, Doris Neumann, Peter Petrovic, Michael Roos, Christoph Vedder

90. Novel Analogues of Bifunctional Ligands for Opioid and Melanocortin 4 Receptor
Vinod V. Kulkarni, Yeon Sun Lee, Christine Salibay, Peg Davis, Shou-wu Ma, Frank Porreca, Victor J. Hruby

91. Fmoc as a Probe in Peptide Purification
Jiangli Song, Zhenchao Gao, Lanlan You, Niansheng Li, XianGang Yang, Wentao Zhang

92. 1,3,5-Triazepan-2,6-diones as Conformationally Constrained Dipeptide Mimetics. In Silico Guided Identification of sPLA2 Inhibitors
Gilles Guichard, Gersande Léna, Joel Boeglin, Pascal Muller, Eric Boilard, Gérard Lambeau, Didier Rognan, Claude Didierjean

93. Proline-based diketopiperazine-scaffolds
Nina Deppermann, Wolfgang Maison

94. Concept and Synthetic Approach for a Kilogram Scale Synthesis of Octa-D-Arginine Amide Nonahydrochloride Salt
J. C. Califano, A. Uribe, J. L. Chang, C. L. Becker, J. J. Napier, V. Kishore, D. Zhou, G. Love, K. Gernhardt, J. C. Tolle

95. Stereoselective Synthesis 0f (3S)- and (3R)-3-Hydroxy-3-(2,6-Dimethyl-4-Hydroxyphenyl)Propanoic Acid and its Incorporation into a Cyclic Enkephalin Analogue
Grazyna Weltrowska, Carole Lemieux, Nga N. Chung, Brian C. Wilkes, Peter W. Schiller

96. Highly Selective Cyclic Hexapeptides Antagonist of GPIIb-IIIa by Multiple N-Methylation
Jayanta Chatterjee, Oded Ovadia, Grit Zahn, Luciana Marinelli, Amnon Hoffman, Horst Kessler

97. Synthesis of N-Boc Protected Hydrazine Diacids as Key Structural Units for the Formation of ±-Helix Mimics
Laura Anderson, Priyesh Jain, Emily McIntosh, Mark L. McLaughlin

98. Solid-Phase Synthesis of 1,3,5-Trisubstituted 1,4-Diazepin-2-one Peptide Mimic
Hassan S. Iden, William D. Lubell

99. General Solid-Phase Phosphopeptide Proteomis with Affinity Pull-Down
Kim Larsen, Kasper K. Sørensen, Steen Gammeltoft, Knud J. Jensen

100. Synthesis and Peptide Coupling of Protected Pyrrolylalanine
Aurélie A. Dörr, William D. Lubell

101. Synthesis of aryl sulfamate and phenol small peptide derivatives using a multidetachable sulfamate linker strategy
Diane Fournier, Pierre-Alain Breuil, Donald Poirier

102. Phe-Aib Hydroxyethylene Dipeptide Isostere Synthesis
Nicolas Genest, Susan Del Valle, Teresa Lama, Willam D. Lubell

103. Poly (vinyl alcohol)-graft-Poly (ethylene glycol) Supported Hydroxyproline: Synthesis and Application in the Enantioselective Aldol Condensation
Tarek Kassem, X. X. Zhu, William D. Lubell

104. Microwave-Assisted Synthesis of Rhodamine Fluorescent Tags
Wajih B. Ben tahar, Jeffrey W. Keillor, William D. Lubell

105. A novel family of diketopiperazines as a tool for the study of transport across the blood-brain barrier (BBB) and their potential use as BBB-shuttles.
Meritxell Teixidó, Esther Zurita, Roger Prades, Teresa Tarrago, Ernest Giralt

106. New Perspective in Peptide Chemistry by N-Alkylation
Horst Kessler, Jayanta Chatterjee, Lucas Doedens, Florian Operrer, Eric Biron, Daniel Hoyer, Herbert Schmid, Chaim Gilon, Victor J. Hruby, Dale F. Mierke

107. Interactions of peptides with single-walled carbon nanotubes
Zhengding Su, Ken Mui, Elisabeth Daub, Tong Leung, John Honek

108. Stimuli-responsive Peptide Self-assembly into Well-organized Nanofibers
Tomoyuki Koga, Ken-ichi Kitamura, Nobuyuki Higashi

109. pH Controlled Aggregation Morphology of Aβ(16–22): Formation of Peptide Nanotubes, Helical Tapes and Amyloid Fibrils
Ronald C. Elgersma, Dirk T. S. Rijkers, Rob M. J. Liskamp

110. Immobilization of Antimicrobial Peptides on Reverse Osmosis Polyamide Membranes: Potential Biofilm Inhibitors?
Karin Berliner, Eyal Hershkovitz, Zeev Ronen, Roni Kasher

111. Synthesis of Polylactides with Side Chain Functionality: Ring-Opening Polymerimerization of a Homobislactone Prepared from Lysine
Hiromi Kodera, Naoki Nishishita, Yoshiaki Hirano, Yoshiaki Kiso, Yoshio Hayashi

112. New Degradable Cationic Peptides for Modulated Gene Delivery
Fiana Mirkin, Hadar Eini, Amos Douvdevani, Gerardo Byk

113. The Dcpm protecting group is a useful alternative to the Hmb residue
Petra Henklein, René Röder, Hardy Weißhoff, Peter Henklein, Louis A. Carpino

114. Development of a RGDS-peptide modified polyurethane for tissue regeneration
A. Rechichi, S. Sartori, A. Caporale, G. Ciardelli, G. Vozzi, L. Mazzucco, E. Peggion, P. Giusti

115. Modulating Collagen Triple-Helix Stability with 4-Chloro, 4-Fluoro, and 4-Methylprolines
Matthew D. Shoulders, Ronald T. Raines

116. Peptide-Chitosan Matrix: a New Multifunctional Biomaterial
Motoyoshi Nomizu, Natsumi Yamagata, Mayumi Mochizuki, Yamato Kikkawa, Yuichi Kadoya

117. Effect of phosphorylation on tau aggregation using model peptides and Circular Dichroism studies
Heather Palmer, Ajoy Basak

118. Peptides for prolonging youth
Marc Heidl

119. The Synthesis of DAMGO-Based Potential Affinity Labels with High Mu Opioid Receptor Affinity and the Formation of Cyclic O-Alkyl Thiocarbamates
Bhaswati Dattachowdhury, Thomas F. Murray, Jane V. Aldrich

120. Amino acid Derivatives of Aporphinic Alkaloid Glaucine and their antioxidant activity
Maya Spasova, Stefan Philipov, Tsenka Milkova

121. Synthesis of Cyclic Tetrapeptide CJ 15,208: A Novel Kappa Opioid Receptor Antagonist
Santosh S. Kulkarni, Nicolette C. Ross, Jay P. McLaughlin, Jane V. Aldrich

122. Exploring the relationship between turn geometry and allosteric antagonism of peptide mimic ligands for the prostaglandin F2α receptor
C. B. Bourguet, X. Hou, S. Chemtob, W. D. Lubell

123. Optimization of the bioconvertion of the Angiotensin I Converting Enzyme inhibitors IPP and VPP
Jos Schalk

124. Tailor made Pharmacokinetics of Peptides by Transient PEGylation
Ulrich Hersel, Martina Kreuzer, Harald Rau, Dirk Vetter, Thomas Wegge

125. Design and Synthesis of Cyclic Arodyn Analogues by Ring-Closing Metathesis (RCM) for Kappa Opioid Receptor (KOP) Antagonists
Wei-Jie Fang, Santosh S. Kulkarni, Thomas F. Murray, Jane V. Aldrich

126. Switch-Peptides as Folding Precursors in Self-Assembling Peptides and Amyloid Fibrillogenesis
M. S. Camus, R. Mimna, A. Schmid, A. Chandravarkar, G. Tuchscherer, H. A. Lashuel, M. Mutter

127. BioShuttle mediated Plasmid Transfer — a Way to new genetic Intervention
Rüdiger Pipkorn, Waldemar Waldeck, Bernd Didinger, Klaus Braun

128. Incorporation of a Novel, Fluorescent and Helicogenic ?-Amino Acid Into Peptaibols: Trichogin Ga IV
C. Baldini, F. Formaggio, C. Toniolo, A. Toffoletti, C. Corvaja, J. -P. Mazaleyrat, K. Wright, J. -F. Lohier, M. Wakselman, B. Orioni, L. Stella, M. Venanzi

129. Seeking for α-Helical Propensity in a Receptor-Bound Conformation of Glucagon-Like Peptide-1
Eunice Murage, Martin Beinborn, Jung-Mo Ahn

130. Conformational Analysis and Folding of Transmembrane and Matrix Peptide Segments of the Mitochondrial Uncoupling Proteins: A Comparative Study
Masoud Jelokhani-Niaraki, Marina V. Ivanova, Cheryl L. Newman, Elizabeth K. Young, Laura Wheaton, Bonnie L. McIntyre, Matthew D. Smith

131. Dynamics study on single and multiple β-sheets
Inta Liepina, Salvador Ventura, Cezary Czaplewski, Adam Liwo

132. Homotrimeric Collagen Peptides As Model Systems For Cell Adhesion Studies
Leslie Barth, Eva K. Sinner, Sergio A. Cadamuro, Christian Renner, Dieter Oesterhelt, Luis Moroder

133. Cyclic Peptide Analogs of Laminin Active Sequences Enhance the Biological Activity
Shu Takaki, Kozue Kato-Takagaki, Nobuharu Suzuki, Shinya Oishi, Yamato Kikkawa, Motoyoshi Nomizu

134. Hydrophobic Peptide Segments in Soluble Proteins Competent For Membrane Insertion: Role in Amyloidogenesis
Fiona Cunningham, Arianna Rath, Charles M Deber

135. Construction and Characterization of Melanocortin-2 and -4 Receptor Chimeras
Krista R Wilson, Bettina Proneth, Hendrik Luesch, Sally A. Litherland, Carrie Haskell-Luevano

136. Expression of Double Transmembrane Domain GPCR Fragments for Biophysical Analysis
Leah S. Cohen, Boris Arshava, Racha Estephan, Jacquelinev Englander, Melinda Hauser, Jeffrey M. Becker, Fred Naider

137. Peptide and Non-Peptide Mimetics Utilize Different Pathways for Signal Transduction
Victor J. Hruby, Minying Cai, Matt Dedek, Hongchang Qu, Erin Palmer, Alexander Mayorov, Dev. Trivedi, George Tsaprailis, Yingqui Yang

138. Structural Studies on Large Fragments of G Protein Coupled Receptors
Fred Naider, Alexey Neumoin, Boris Arshava, Leah S. Cohen, Jeffrey M. Becker, Oliver Zerbe

139. Isolation of the Influenza A HA2 C-terminal segment by combination of nonionic detergents
Yulia A. Smirnova, Natalya V. Fedorova, Aleksander L. Ksenofontov, Larisa V. Kordyukova, Marina V. Serebryakova, Ludmila A. Baratova, Boris V. Vaskovsky

140. Molecular Imaging and Orientational Changes of Antimicrobial Peptides in Membranes
Tzong-Hsien Lee, Kristopher Hall, Adam Mechler, Lisandra Martin, Jonathan Popplewell, Gerry Ronan, Marie-Isabel Aguilar

141. Glycated-CD59 antigen: exploration of synthetic approaches
S. Cantel, A. Kavishwar, M. Schlimme, A. Khatri, J. A. Halperin, M. Chorev

142. A combination of ligand SAR and receptor site-directed mutagenesis reveals requirements for antagonist activity at the melanocortin-3 receptor
Bettina Proneth, Federico P. Portillo, Carrie Haskell-Luevano

143. Conformational Effects of Cyclic Hexapeptides for Ion Channel Properties
Junichi Taira, Satoko Imamura, Satoshi Osada, Masoud Jelokhani-Niaraki, Tsuguhisa Ehara, Hiroaki Kodama

144. Synthesis and Biological Activities of Cyclic Peptide, Hymenamide Analogs
Yasuhiro Shiki, Mika Onai, Daisuke Sugiyama, Satoshi Osada, Ichiro Fujita, Hiroaki Kodama

145. Monitoring Glucagon and Glucagon Antagonist-Mediated Internalization: A Useful Approach to Study Glucagon Receptor Pharmacology
Pallavi Sachdev, Laxmi Manohar Tirunagari, Dennis Kappei, Cecilia G. Unson

146. Semi-Synthetic Strategies to Obtain Glucosylated MOG to Identify Antibodies as Biomarkers in Multiple Sclerosis Disease
Francesca Gori, Barbara Mulinacci, Eva Bonchi, Mario Chelli, Francesco Lolli, Anna M. Papini, Paolo Rovero

147. Photoprobe Peptides to Map the Interactions of Angiotensin II with its Receptor AT1

D. Fillion, G. Guillemette, R. Leduc, E. Escher

148. Synthesis and Biological Activity of Transmembrane Peptides Derived from FPR Family Receptors
Daisuke Sugiyama, Ryo Hayashi, Satoshi Osada, Yuhei Hamasaki, Ichiro Fujita, Hiroaki Kodama

149. Incorporation of the Unnatural Amino Acid p-benzoyl-L-phenylalanine (Bpa) into a G Protein-coupled Receptor in its Native Context
George Umanah, Li-Yin Huang, Peter G. Schultz, Fred Naider, Jeffrey M. Becker

150. Ion Channel Formation of Dimeric Peptide Enhanced by Electrostatic Inter-Helical Interactions
Junichi Taira, Satoshi Osada, Masoud Jelokhani-Niaraki, Tsuguhisa Ehara, Hiroaki Kodama

151. Temperature-induced Ligand Contact Point Variations of the hAT1 Receptor and of the Constitutively Active Mutant N111G-hAT1

J. Arsenault, M. P. La-Haye Renaud, M. Clément, D. Fillion, G. Guillemette, R. Leduc, P. Lavigne, E. Escher

152. Structural changes in the binding pocket of the liganded angiotensin II receptor AT1 during activation.
Martin Clément, Gaétan Guillemette, Richard Leduc, Emanuel Escher

153. Vaccine delivery utilizing liposaccharides
Pavla Simerska, Ross P. McGeary, Abu-Baker M. Abdel-Aal, Peter M. Moyle, Colleen Olive, Michael F. Good, Istvan Toth

154. Vaccine Delivery: Synthesis and Investigation of a Highly Pure, Multi-Epitopic Lipopeptide Vaccine Candidate
Istvan Toth, Peter M. Moyle, Pavla Simerska, Yoshio Fujita, Colleen Olive, Michael F. Good

155. Synthesis of Mannosylated Glycopeptides as Components for Synthetic Vaccines
Renata Kowalczyk, Margaret A. Brimble, Rod Dunbar

156. Bradykinin Analogues Acylated On Their N-terminus — Some Recent Development
Dariusz Sobolewski, Adam Prahl

157. Rationally-designed Multivalent Architectures for Mimicking Homotrimers of CD40L, a Member of the TNF Superfamily
Gilles Guichard, Nathalie Trouche, Sébastien Wieckowski, Weimin Sun, Olivier Chaloin, Alberto Bianco, Johan Hoebeke, Pascal Schneider, Sylvie Fournel

158. A Strategy for Selectively Shielding Portions of a Peptide/Protein from Immune Response while Maintaining Immunogenicity of Contiguous Epitopes
Elisabetta Bianchi, Marco Finotto, Paolo Ingallinella, Mike Citron, Renee Hrin, Meiqing Lu, Romas Geleziunas, Michael D. Miller, Xiaoping Liang, Antonello Pessi

159. Synthesis of Peptide-Based Vaccines
Zhanna Potetinova, Gordon E. Willick

160. A Peptide Vaccine Based on Retro-Inverso β-Amyloid Sequences Fails to Elicit a Cross-reactive Immune response
Elisabetta Bianchi, Paolo Ingallinella, Marco Finotto, Xiaoping Liang, Gene G. Kinney, Antonello Pessi

161. Synthesis and Application of (Z)-Alkene- and (E)-Fluoroalkene-Dipeptide Isosteres as cis-Amide Equivalents
Kenji Tomita, Tetsuo Narumi, Ayumu Niida, ya Oishi, Hiroaki Ohno, Nobutaka Fujii

162. Gadd45β dimerization does not affect MKK7 binding
Laura Tornatore, Simona M. Monti, Daniela Marasco, Nina Dathan, Rosa M. Vitale, Ettore Benedetti, Carlo Pedone, Salvatore Papa, Guido Franzoso, Menotti Ruvo

163. A Glycopeptide-based Technique for Selective Antibody Purification
Elisa Peroni, Marta Tontini, Barbara Mulinacci, Mario Chelli, Francesco Lolli, Paolo Rovero, Anna M. Papini

164. C-Terminal Amidation On Aryl Hydrazine Resin
Witold A. Neugebauer, Amélie Parent, Xue Wen Yuan, Robert Day

165. Synergy Between a Lead Proline-rich Antibacterial Peptide Derivative and Small Molecule Antibiotics
Laszlo Jr Otvos, Marco Cassone, Vanessa de Olivier Inacio, Paul Noto, John J. Rux, John D. Wade, Predrag Cudic

166. Natural mutants of HIV CTL epitopes with enhanced immunogenicity as potential vaccine candidates
Sylvie E. Blondelle, Rosa Moya, Kim Schroder, Keiko Osawa, Darcy B. Wilson

167. Lipodepsipeptide antibiotic fusaricidin and its analogues. Total solid-phase and biological activity.
Maciej Stawikowski, Pedrag Cudic

168. Progress toward Total Solid-Phase Synthesis of Depsipeptide Antibiotic Katanosin B
Roma Stawikowska, Maciej Stawikowski, Predrag Cudic

169. Determination of the minimal fusion peptide of HIV, SIV and BLV fusion glycoproteins
Aurélien Lorin, Benoît Charloteaux, Laurence Lins, Vincent Stroobant, Robert Brasseur

170. Development of a Novel Fusion Inhibitor against T-20-resistant HIV-1
Shinya Oishi, Saori Ito, Hiroki Nishikawa, Michinori Tanaka, Hiroaki Ohno, Akira Otaka, Kazuki Izumi, Eiichi Kodama, Masao Matsuoka, Nobutaka Fujii

171. ε-Peptide Chimeras as Novel Antimicrobials
Yi-An Lu, Jin-Long Yang, James P. Tam

172. Chemical modifications of short antimicrobial peptides from insects and vertebrates to fight multi-drug resistant bacteria
Daniel Knappe, Christin Stegemann, Ariane Nimptsch, Alexander Jr Kolobov, Ekaterina Korableva, Olga Shamova, Vladimir N. Kokryakov, Ralf Hoffmann

173. Isolation of Peptides From Rat Tissues: Peptidomics vs. Degradomics
Oleg N. Yatskin, Olga V. Sazonova, Dmitry P. Khachin, Elena Y. Blishchenko, Andrei A. Karelin, Vadim T. Ivanov

174. Multivalent peptidomimetics for tumor targeting
Nadine Pannier, Valerie Humblet, Preeti Misra, John Frangioni V., Wolfgang Maison

175. Comparison of [18F]FBA and [18F]FPyMe as peptide radio-labeling agents of PEPHC1 for PET imaging of EGFRvIII
Charlotte L. Hansen, Bertrand Kuhnast, Franciose Hinnen, Frédéric Dollé, Nic Gillings, Paul R. Hansen, Andreas Kjær

176. Carbohydrated [99mTc(CO)3](NαHis)Ac-Bombesin(7–14) analogs
Veronique Maes, Luc Brans, Christian Schweinsberg, Elisa Garcia-Garayoa, Peter Bläuenstein, Peter A. Schubiger, Dirk Tourwé

177. A Synthetic Peptide Approach for Elucidating the Points of Natural Auto-Antibody Reactivity to Proteolytic Fragments of Human IgG
A. Schmidt, D. De Riggi, R. E. Jordan, B. Whitaker, G. A. Heavner, M. Kruszynski

178. Heterobivalent Ligands Crosslink Multiple Cell-Surface Receptors — A Step Towards Personal Medicine
Jatinder S. Josan, Rajesh Sankaranarayanan, Heather L. Hand, Steve Fernandes, Liping Xu, Josef Vagner, Robert J. Gillies, Victor J. Hruby

179. Development of Polyvalent Peptide-Conjugated Magnetic Nanoparticles for Targeted In-Vivo Imaging of Micro-Thrombi
Rana Filfil, Albert Jin, Dmitri Tolkatchev, Kenji Tonan, Richard Gingras, Philip A. Barber, Feng Ni

180. Design, Selection and Binding Mechanism of Bivalent Miniproteins Targeting Human Thrombin
Andy Ng, Jamshid Tanha, Saran Narang, Feng Ni

181. Quenched Fluorescent Peptide Substrates as Tools for the Discovery of Novel Cardiovascular Disease Biomarkers
A. Ian Smith, Fiona J. Warner, Rebecca A. Lew, Mike Yarski, Barry McGrath, Louise M. Burrell

182. Solid Phase Synthesis and Analysis of Amadori Peptides
Andrej Frolov, David Singer, Thomas Zauner, Ralf Hoffmann

183. Design of Hetero-Bivalent Polypeptides as Kinetics-Based Sensors for High-Sensitivity Detection of Weak Molecular Interactions
Kenji Tonan, Dmitri Tolkatchev, Ping Xu, Ping Wang, Josee Plamondon, Anna Vinogradova, Richard Gingras, Feng Ni

184. Monitoring of native chemical ligation by surface plasmon resonance
Ewa Wieczerzak, Raymond Jr Hamel, Vincent Chabot, Vincent Aimez, Paul G. Charette, Michel Grandbois, Emanuel Escher

185. Studies for Identification of the Minimal Epitope(s) mimicked by the Synthetic Glucopeptide CSF114(Glc)
Francesca Nuti, Barbara Mulinacci, Elisa Peroni, Maria C. Alcaro, Ilaria Paolini, Francesco Benedetti, Alfonso Carotenuto, Francis Ciolli, Francesco Lolli, Mario Chelli, Paolo Rovero, Anna M. Papini

186. Synthesis of Bivalent MSH Ligands and Evaluation of their Binding to hMC4R using MSH Lanthaligand
Steve M. Fernandes, Rajesh Sankaranarayanan, Liping Xu, Jatinder Josan, Josef Vagner, Robert Gillies, Victor J. Hruby

187. Synthesis Of Organometallic Glycopeptides And Electrochemical Studies To Detect Autoantibodies In Multiple Sclerosis Patients'Sera.
Feliciana Real-Fernández, Amélie Chamois-Colson, Jérome Bayardon, Francesca Nuti, Elisa Peroni, Maria R. Moncelli, Rita Meunier-Prest, Sylvain Jugè, Anna Maria Papini

188. Tumor Imaging With Tetrabranched Neurotensin
Monica Fabbrini, Chiara Falciani, Barbara Lelli, Alessandra Cappelli, Alessandro Pini, Luisa Lozzi, Luisa Bracci

189. A new and selective radiolabeled αVβ3 peptide antagonist as tracer in tumor diagnosis
Stefania De Luca, Annarita Del Gatto, Menotti Ruvo, Maria Rosaria Panico, Antonella Zannetti, Silvana Del Vecchioiano, Marco Salvatore, Carlo Pedone, Michele Saviano, Laura Zaccaro

190. Ribose Building Block For The Synthesis Of Glycopeptides For Fishing Out Antibodies In Autoimmune Diseases
Ma Angeles Bonache, Alexandra Le Chevalier, Francesca Nuti, Elisa Peroni, Mario Chelli, Paolo Rovero, Anna M. Papini

191. Design, Synthesis and Pharmacological Characterization of Fluorescein-Derived Endothelin Antagonists Bq-123 And Bq-788
Jean-Philippe Brosseau, Witold A. Neugebauer, Fernand Jr Gobeil, Pedro D'Orléans-Juste

192. Peptide Antagonists of the PED-hPLD1 Binding
F. Viparelli, N. Doti, S.M. Monti, D. Marasco, N. Dathan, C. Pedone, C. Miele, P. Formisano, F. Beguinot, M. Ruvo

193.
In vivo Imaging Using Tissue Specific Near Infrared fluorescent Peptide Conjugate, c[RGDyK(HiLyte Fluor™ 750)]
Jose I. Rey, Haihong Huang, Ling Sheng, Xiao Fen Zhong, Rich Meyer, Xiaohe Tong, Francis Moussy, Anita Hong

194. Photoinduced Intramolecular Covalent Bond Formation in Structurally Rigid -Bpa-(spacer)-Met Hexapeptides
Alessandro Moretto, Simona Oancea, Fernando Formaggio, Claudio Toniolo, Laurence A. Huck, Dino Mangion, William J. Leigh

195. Evaluation of chemically and enzymatically prepared cross-linked BNP fragments
Ganga Beligere, Huaiqin Wu, Jim Fino, Reika Campbell

196. Monitoring of MMPs activity in vivo, non-invasively, using solubility switchable MRI contrast agent
Beata Jastrzebska, Rejean Lebel, Oliver J. McIntyre, Benoit Paquette, Witold Neugebauer, Emanuel Escher, Martin Lepage

197.
99mTc-labeled Ac-DEVD Peptides as a Substrate for Measuring Caspase Activity
Chiyi Xiong, Zhi Yang, Rui Zhang, William Tong, Juri Gelovani, Chun Li

198. PepLook: An innovative in silico tool for determination of structure, polymorphism and stability of peptides
Annick Thomas, Sébastien Deshayes, Marc Decaffmeyer, Marie-Hélène Van Eyck, Benoit Charloteaux B, Robert Brasseur

199. The Effects of the EW — Peptide Optical and Chemical Isomers on the Hemopoietic Stem Cells in Intact and Irradiated Mice
Vladislav I. Deigin, Tamara N. Semenets, Irina A. Zamulaeva, Yana V. Maliutina, Elena I. Selivanova, Alexander S. Saenko, Olga V. Semina

200. N-(Fluorenyl-9-methoxycarbonyl)amino Acid Amide Derivatives as a New Class of Anti-cancer Agents
Lajos Gera, Daniel C. Chan, Vitalija Simkeviciene, Paul A. Jr Bunn, John M. Stewart

201. Opportunities and Challenges of Developing Peptide Drugs in the Pharmaceutical Industry
Waleed Danho, Joseph Swistok, Wajiha Khan, Xin-Jie Chu, Adrian Cheung, David Fry, Hongmao Sun, Grazyna Kurylko, Leonid Rumennik, Joseph Cefalu, Gretchen Cefalu, Philip Nunn

202. Inhibition of pathogenically-related morphologic transition in Candida albicans by disrupting Cdc42 binding to its effectors
Hongjian Li, Yang Li, Feng N, Zhengding Su

203. Synthesis and Pharmacological Evaluation of Highly Potent [Dmt1]DALDA Analogs
P. Anantha Reddy, Anita H. Lewin, Peter W. Schiller

204. Protease-resistant glucagon like peptide-1 analogs with long-term anti-diabetes type 2 activity
Hongjian Li, Cindy X Zhou, Zhengding Su

205. The discovery and development of a natural combinatorial peptide template: the cyclotides
David C. Ireland, Michelle L. Colgrave, Norelle L. Daly, David J. Craik

206. Cyclic peptides as VEGF receptor antagonist
Victor Goncalves, Benoit Gautier, Christiane Garbay, Michel Vidal, Nicolas Inguimbert

207. Facile Synthesis of Hydrocarbon-Stapled Peptides

208. Isolation of angiotensin I converting enzyme inhibitory peptides from a fish by-products hydrolysate Tensideal®
Véronique Lahogue, Karine Vallée-Rehel, Mylène Cuart, Dominique Haras, Patrick Allaume

209. Novel Melanocortin-4 Receptor Agonists That Decrease Food Intake and Body Weight
Jesse Z. Dong, Daniel B. DeOliveira, Heather A. Halem, John E. Taylor, Pierre Roubert, Pascale Plas, Michael D. Culler, Jundong Zhang

210. GHS-1a Agonists That Effectively Stimulate Food Intake and Body Weight Gain
Jesse Z. Dong, Jundong Zhang, John E. Taylor, Heather A. Halem, Rakesh Datta, Michael D. Culler, John Eynon

211. Conformation-activity relationships of cyclo-constrained μ/5 opioid agonists derived from the N-terminal tetrapeptide segment of dermorphin/deltorphin
Jerzy Ciarkowski, Cezary Czaplewski, Sylwia Luczak, Sylwia Rodziewicz-Motowidlo, Irena Berezowska, Peter W. Schiller

212. Deltorphin analogs restricted via a urea bridge: structure and opioid activity
J. Ciarkowski, A. Zieleniak, S. Rodziewicz-Motowidlo, Ł Rusak, N.N. Chung, C. Czaplewski, E. Witkowska, P. W. Schiller, J. Izdebski

213. Synthesis and Characterization of Dimeric Venom Peptides
J. Vizzavona, A. Zufferey, K. Rose

214. Glycosyl-Enkephalins: Synthesis and Binding at the Mu, Delta & Kappa Opioid Receptors. Antinociception in Mice
Charles M. Keyari, Brian I. Knapp, Jean M. Bidlack, John Lowey, Edward J. Bilsky, Robin Polt

215. Agonists and Partial Antagonists Acting on the Leptin—Leptin Receptor Interface
Laszlo Otvos, Marco Cassone, Marianna Terrasi, Sandra Cascio, George D. Mateo, Daniel Knappe, Ralf Hoffmann, Predrag Cudic, John D. Wade, Eva Surmacz

216. Effect of 4-Fluoro-L-proline on the SH3 Binding Affinity
Paolo Ruzza, Chiara Rubini, Giuliano Siligardi, Rohanah Hussain, Andrea Calderan, Andrea Guiotto, Luca Cesaro, Anna M. Brunati, Arianna Donella-Deana

217. Analogues of arginine vasopressin modified in the N-terminal part of the molecule with pipecolic acid isomers
Dariusz Sobolewski, Adam Prahl, Jiřina Slaninová, Bernard Lammek

218. Analogues of arginine vasopressin modified at position 2 with proline derivatives: selective antagonists of oxytocin in vitro

Dariusz Sobolewski, Adam Prahl, Jiřina Slaninová, Bernard Lammek

219. Multimeric peptides as agonists of the erythropoietin receptor
Oscar Vadas, Keith Rose

220. Synthesis and in vitro Pharmacological Profile of Potent and Selective Peptidic V1a Receptor Agonists.
Kazimierz Wisniewski, Robert Galyean, Hiroe Taki, Sudar Alagarsamy, Glenn Croston, Regent Laporte, Claudio D. Schteingart, Pierre J-M. Rivière

221. Discovery of a Ligand that Compensates for Decreased Endogenous Agonist Potency of Melanocortin-4 Receptor Polymorphisms Identified in Obese Humans
Carrie Haskell-Luevano, Zhimin Xiang, Andrzej M. Wilczynski, Kimberly R. Haskell, Amy M. Andreasen, Sally A. Litherland, William J. Millard, Ira D. Pogozheva, Henry I. Mosberg, Nicholas B. Sorenson

222. High-affinity FGFR2 Binding Peptides Derived from the Native Epitope of the KGF Ligand
Yijun Pan, Yvonne M. Angell, Jennifer M. Green, Kathy L. Wright, Joy Miguel, Peter J. Schatz, Christopher P. Holmes

223. Application of Intramolecular Migration Reaction in Peptide Chemistry to Chemical Biology, Chemical Pharmaceutics and Medicinal Chemistry
Yoshio Hayashi, Yuri Yamazaki, Mariusz Skwarczynski, Youhei Sohma, Atsuhiko Taniguchi, Mayo Noguchi, Tooru Kimura, Saskia Neuteboom, Barbara Potts, G. Kenneth Lloyd, Yoshiaki Kiso

224. Synthesis & Biological Evaluation of PYY(3–36) Analogs Substituted with Alanine
John S. Ahn, Ramina Nazarbaghi, Lawrence J. D'Souza, Soumitra Ghosh, Carolyn M. Jodka, Aung N. Lwin, Odile E. Levy

225. Development of μ/δ Opioid Ligands: Enkephalin Analogues Containing 4-Anilidopiperidine Moiety
YeonSun Lee, Ravil Petrov, Vinod Kulkarni, Byoung J. Min, Shou-wu Ma, Peg Davis, Janice Oyarzo, Todd Vanderah, Josephine Lai, Frank Porreca, Ruben Vardanyan, Victor J. Hruby

226. Factors that Affect Dissociation Degree of Strong Aggregated Peptide Chains when Bound to a Polymer or Free in Solution
Luciana Malavolta, Clóvis R. Nakaie

227. Development of AEZS-115 (ZEN-019) by Optimization of Structurally Unique, Orally Active, Peptidomimetic GnRH Antagonists
K. W. Paulini, S. Baasner, M. Gerlach, E. E. Polymeropoulos, P. Schmidt, T. Schuster, M. Teifel, E. G. Guenther

228. Synthesis and solid-phase application of suitably protected γ-hydroxyvaline building blocks
Mare Cudic, Frank Marí, Gregg B. Fields

229. Synthesis and Structure-based Dissection of Cyclic Peptide Chitinase Inhibitors: New Leads for Antifungal and Anti-Inflammatory Drugs
Mark J. Dixon, Amit Nathubhai, Ole A. Andersen, Daan M. F. van Aalten, Ian M. Eggleston

230. Synthesis of Biotin-Tagged Diketopiperazine-Based Anti-Microtubule Agents and Tubulin Photoaffinity Labeling
Yuri Yamazaki, Kyoko Kohno, Hiroyuki Yasui, Yoshiaki Kiso, Saskia Neuteboom, Ana M. Barral, Barbara Potts, G. Kenneth Lloyd, Yoshio Hayashi

231. Study on Interactions of Oligo(tyrosine sulfate)s with Synthetic Heparin-binding Peptides by Affinity Chromatography and MALDI-TOF-MS
Miyuki Yamaguchi, Masaaki Ueki

232. Fallaxin analogues with improved antibacterial activity
S. L. Nielsen, N. Frimodt-Møller, P. R. Hansen

233. Alkene/Alkane-Bridged Mimics of the Lantibiotic Nisin: Toward Novel Peptide-Based Antibiotics
Rianne A. G. Harmsen, Nourdin Ghalit, Johan Kemmink, Hans W. Hilbers, Eefjan Breukink, Dirk T. S. Rijkers, Rob M. J. Liskamp

234. Peptide-Lisinopril Conjugates: Design, Synthesis and Biological Activities
Josue Alfaro-Lopez, Chris Soares, Soumitra Ghosh, Alexander Kravchuk, Eugene Coates, Lynn Jodka, Amy Carroll, Que Liu

235. Novel Bifunctional Peptides as Opioid Agonists and NK-1 Antagonists
Padma Nair, Takashi Yamamoto, Vinod Kulkarni, Sharif Moye, Edita Navratilova, Peg Davis, Tally Largent, Shou-wu Ma, Henry I. Yamamura, Todd Vanderah, Josephine Lai, Frank Porreca, Victor J. Hruby

236. Anti-HIV dendrimeric peptides
Qitao Yu, Ling Li, James P. Tam

237. Ago-Antagonists for G Protein-Coupled Peptide Hormone Receptor by Modifying the Agonist's Signalling Domain
Michael Beyermann, Nadja Heinrich, Klaus Fechner, Jens Furkert, Wei Zhang, Oliver Kraetke, Michael Bienert, Hartmut Berger

238. Model of Intermolecular Interactions between High Affinity Phosphopeptides and Stat3
John S. McMurray, Zhiyong Ren, Pijus K. Mandal, Xiaomin Chen

239. Inhibition of Stat3 by Cell-Permeable Peptidomimetic Prodrugs Targeted to its SH2 Domain
John S. McMurray, Pijus K. Mandal, Warren S. Liao, Zhiyong Ren, Xiaomin Chen

240. Synthesis and Biological Activity of Conformational Restricted Galanin Fragments
Marcus Marra, Marcos A. Fázio, Antonio Miranda

241. Interaction of membrane mimetic vesicles with the antimicrobial peptide gomesin and its analogues
Marcela S. Carmona, Luis G. M. Moraes, Marcos A. Fázio, Rosemaire A. S. Lucca, Maria L. V. Oliva, Sirlei Daffre, Antonio Miranda

242. Limited Structure-Activity Relationships for Carboxy and AminoTerminal Substitutions of Peptide YY 25–36
David H. Singleton, James G. Boyd, Nancy A. Nardone, Brett S. Robinson, Lydia C. Pan, John R. Hadcock, A. Zane Wenzel

243. Cysteine Based PNA (CPNA): Design and Synthesis of Novel CPNA Monomers
Sung Wook Yi, Priyesh Jain, Mehul Ajmera, Sridhar Reddi Kaulagari, Melissa Topper, Laura Anderson, Mark L. McLaughlin

244. Synthesis and Biological Activity of Nicotianamine and Analogues
M'Barek Bouazaoui, St é phane Mari, Pierre Czernic, Catherine Curie, Jean Martinez, Florine Cavelier

245. The active site specificity of angiotensin II converting enzyme 2 investigated through single and multiple residue changes and β-amino acid substrate analogs.
Daniel Clayton, Iresha Hanchapola, Patrick Perlmutter, A. Ian Smith, Marie-Isabel Aguilar

246. Effects of net charge and the number of positively charged residues on the biological activity of amphipathic α-helical cationic antimicrobial peptides
Ziqing Jiang, Adriana I. Vasil, John Hale, Robert E. W. Hancock, Michael L. Vasil, Robert S. Hodges

247. Action of Bauhinia-derivated compounds on Callosobruchus maculatus development
Joana T. Sumikawa, Marlon V. Brito, Ana Paula U. Araújo, Maria Ligia R. Macedo, Maria Luiza V. Oliva, Antonio Miranda

248. Positively charged gramicidin A based peptides form two types of membrane channels
Sergey I. Kovalchuk, Elena A. Kotova, Tatyana B. Stoilova, Sergey V. Sychev, Natalya S. Egorova, Andrey Y. Surovoy, Yuri N. Antonenko, Vadim T. Ivanov

249. Effects of Tumor-Associated Mutations in the p53 Tetramerization Domain on Oligomerization State and Transcriptional Activity
Rui Kamada, Tomoko Terai, Takao Nomura, Yoshiro Chuman, Toshiaki Imagawa, Kazuyasu Sakaguchi

250. Self-association regions in the CARD of Bcl-10
M. Ruvo, A. Sandomenico, D. Marasco, S. M. Monti, B. Tizzano, A. De Capua, C. Pedone, A. Saporito, R. M. Vitale, S. Formisano, R. Stilo, D. Liguoro

251. GHRP-2 Attenuates Burn-Induced Dysfunctions in Rodents
Ambikaipakan Balasubramaniam, Rashika Joshi, Lou Ann Friend, J. Howard James

252. Peptides binding the type E immunoglobulins
Annamaria Sandomenico, Daniela Marasco, Simona M. Monti, Michele Saviano, Carlo Pedone, Ettore Benedetti, Menotti Ruvo

253. Evolution of the Synthetic Process to Prepare the Tripeptide Segment of ABT-510
Calvin L. Becker, Jean Christophe Califano, John C. Tolle, James J. Napier, Lawrence Kolaczkowski, Sou-Jen Chang, Zhenping Tian, Sukamar Manna

254. Retrocyclin-2: a potent anti-HIV θ-defensin that forms a cyclic cystine ladder structural motif
Norelle L. Daly, Chen K. Yi, Johan K. Rosengren, Ute C. Marx, Martin L. Phillips, Alan J. Waring, Wei Wang, Robert I. Lehrer, David J. Craik

255. Isothermal Titration Calorimetry and Inhibition of Platelets Aggregation by [D-Phe/(Transcinnamoyl)-Pro-D-Arg-P1'-CONH2] Peptides Inhibitors of Thrombin
Cristina C. Clement, Anna Babinska, Elizabeth Kornecki, Manfred Philipp

256. Trypsin Stability of Lysine-Peptoid Hybrids
Trine S. Ryge, Paul R. Hansen

257. A Comparative Examination of two Fmoc Removal Reagents for Process Improvement to Produce Peptide Drugs
K. Srivastava, Davis M.

258. Bicyclic Organo-Peptides as Models for Carbohydrate Binding Proteins
Claudia James-Johnson, Predrag Cudic

259. Impurity Rejection in the Crystallization of ABT-510 as a Method to Establish Starting Material Specifications
John C. Tolle, Calvin L. Becker, Jean C. Califano, Jane L. Chang, Kevin Gernhardt, James J. Napier, Steven J. Wittenberger, Judy Yuan

260. Spatially Defined Peptide-Polymer Biotherapeutic Synthesis on Novel Cross-linked Beads with ‘Spatially Tunable’ and ‘Isolated’ Functional Sites
M.K. Jacob, K.S. Kumar

261. Supramolecular Aggregates derivatized by CCK8 Peptide as Selective Nanocarriers for Drug Delivery
Antonella Accardo, Diego Tesauro, Giancarlo Morelli, Luigi Del Pozzo, Carlo Pedone, Anna Lucia Tornesello, Ettore Benedetti

262. The role of Cell Penetrating Peptides (CPPs) in membrane lipid phase behavior: a novel aspect elucidating peptide-mediated delivery
Cinzia Esposito, AiWei Tian, Mario Scrima, Karolina Kieres, Pietro Campiglia, Anna Maria D'Ursi, Tobias Baumgart

263. Factors that influence oral bioavailability; A cathepsin K inhibitor for human studies
Daniel F. Veber

264. Injectable Biodegradable Polymer Depots For Minimally Invasive Delivery of Peptides and Proteins
Li Zhang, Steven P. Schwendeman

Keywords: Chemistry, Medicinal Chemistry, Medical Microbiology, Proteomics, Immunology

Author(s)
 
 
Publisher
Springer
Publication year
2009
Language
en
Edition
1
Series
Advances in Experimental Medicine and Biology
Page amount
746 pages
Category
Natural Sciences
Format
Ebook
eISBN (PDF)
9780387736570

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